Highly selective and orally active non-peptide endothelin-A (ETA) receptor antagonist with IC50 values of 0.3 nM for ETA and 480 nM for ETB receptors, indicating potent selectivity.
Effective antihypertensive agent that inhibits ET-1-induced pressor responses when administered orally, showcasing its potential in cardiovascular research and therapeutic applications.
Available in a 10 mg pack, this HPLC grade >98% purity reagent is essential for precise biochemical assays and research.
